Structurally the Center for Drug Chemistry includes two chemical laboratories (laboratory of synthesis #1 and laboratory of synthesis #2), three biological laboratories (pharmacology, chemotherapy of infectious diseases and toxicology), a section on pharmacokinetics, animal facilities, an analytical chemisitry department with a group of physical methods, department of development of forms of medicinal preparations, a department of industrial technology, a department or research organization, scientific library and auxiliary subdivisions.

The laboratories and departments of Institute are specially designed for research and experimental work and are equipped with the necessary research facilities.

General Director of the Center for Drug Chemistry - Robert Glushkov, D.Sc., Professor, Member of Russian Academy of Medical Sciences, Merited Scientist, Winner of State Prize of USSR and Prize of Ministry Council of USSR.